PROJECT OUTPUTS

RECENT ENOCH SCIENTIFIC PUBLICATIONS

2020

BALIK, V. AND K. TAKIZAWA Safe and bloodless exposure of the third segment of the vertebral artery: a step-by-step overview based on over 50 personal cases. Neurosurgical Review, Dec 2019, 42(4), 991-997.
Q2

BORKOVA, L., I. FRYDRYCH, N. JAKUBCOVA, R. ADAMEK, et al. Synthesis and biological evaluation of triterpenoid thiazoles derived from betulonic acid, dihydrobetulonic acid, and ursonic acid. European Journal of Medicinal Chemistry, Jan 2020, 185, 18.
T10

GRUNER, B., J. BRYNDA, V. DAS, V. SICHA, et al. Metallacarborane Sulfamides: Unconventional, Specific, and Highly Selective Inhibitors of Carbonic Anhydrase IX. Journal of Medicinal Chemistry, Nov 2019, 62(21), 9560-9575.
T5

HODON, J., L. BORKOVA, J. POKORNY, A. KAZAKOVA, et al. Design and synthesis of pentacyclic triterpene conjugates and their use in medicinal research. European Journal of Medicinal Chemistry, Nov 2019, 182, 25.
T10

KAEOPOOKUM, P., M. PETRIK, D. SUMMER, M. KLINGER, et al. Comparison of Ga-68-labeled RGD mono- and multimers based on a clickable siderophore-based scaffold. Nuclear Medicine and Biology, Nov-Dec 2019, 78-79, 1-10.
Q2

LIGASOVA, A., M. VYDRZALOVA, R. BURIANOVA, L. BRUCKOVA, et al. A New Sensitive Method for the Detection of Mycoplasmas Using Fluorescence Microscopy. Cells, Dec 2019, 8(12), 17.
Q1

MAZURENKO, S., Z. PROKOP AND J. DAMBORSKY Machine Learning in Enzyme Engineering. Acs Catalysis, Jan 2020, 10(2), 1210-1223.
T10

PERLIKOVA, P., M. KVASNICA, M. URBAN, M. HAJDUCH, et al. 2-Deoxyglycoside Conjugates of Lupane Triterpenoids with High Cytotoxic Activity-Synthesis, Activity, and Pharmacokinetic Profile. Bioconjugate Chemistry, Nov 2019, 30(11), 2844-2858.
Q1

VAVRA, O., J. FILIPOVIC, J. PLHAK, D. BEDNAR, et al. CaverDock: a molecular docking-based tool to analyse ligand transport through protein tunnels and channels. Bioinformatics, Dec 2019, 35(23), 4986-4993.
Q1

VOLLER, J., T. BERES, M. ZATLOUKAL, P. DZUBAK, et al. Anti-cancer activities of cytokinin ribosides. Phytochemistry Reviews, Aug 2019, 18(4), 1101-1113.
T10

2019

CAPKOVA, Z., P. CAPKOVA, J. SROVNAL, K. STAFFOVA, et al. Differences in the importance of microcephaly, dysmorphism, and epilepsy in the detection of pathogenic CNVs in ID and ASD patients. Peerj, Nov 2019, 7, 17.
Q2

JORDA, R., E. REZNICKOVA, U. KIELCZEWSKA, J. MAJ, et al. Synthesis of novel galeterone derivatives and evaluation of their in vitro activity against prostate cancer cell lines. European Journal of Medicinal Chemistry, Oct 2019, 179, 483-492.
T10

KADLECOVA, A., B. MAKOVA, M. ARTAL-SANZ, M. STRNAD, et al. The plant hormone kinetin in disease therapy and healthy aging. Ageing Research Reviews, Nov 2019, 55, 12.
T10

KOKKONEN, P., D. BEDNAR, G. PINTO, Z. PROKOP, et al. Engineering enzyme access tunnels. Biotechnology Advances, Nov 2019, 37(6), 13.
T5

MILISIUNAITE, V., A. KADLECOVA, A. ZUKAUSKAITE, K. DOLEZAL, et al. Synthesis and anthelmintic activity of benzopyrano 2,3-c pyrazol-4(2H)-one derivatives. Molecular Diversity, 18.
Q3

NOWIKOW, C., R. FUERST, M. KAUDERER, C. DANK, et al. Synthesis and biological evaluation of cis-restrained carbocyclic combretastatin A-4 analogs: Influence of the ring size and saturation on cytotoxic properties. Bioorganic & Medicinal Chemistry, Oct 2019, 27(19), 13.
Q2

VANDA, D., P. ZAJDEL AND M. SOURAL Imidazopyridine-based selective and multifunctional ligands of biological targets associated with psychiatric and neurodegenerative diseases. European Journal of Medicinal Chemistry, Nov 2019, 181, 25.
T10

BURYSKA, T., M. VASINA, F. GIELEN, P. VANACEK, et al. Controlled Oil/Water Partitioning of Hydrophobic Substrates Extending the Bioanalytical Applications of Droplet-Based Microfluidics. Analytical Chemistry, Aug 2019, 91(15), 10008-10015.
T10

JORDA, R., S. M. M. LOPES, E. REZNICKOVA, H. AJANI, et al. Tetrahydropyrazolo 1,5-a pyridine-fused steroids and their in vitro biological evaluation in prostate cancer. European Journal of Medicinal Chemistry, Sep 2019, 178, 168-176.
T10

VOLODKO, N., T. GUTOR, O. PETRONCHAK, R. HULEY, et al. Low infiltration of tumor-associated macrophages in high c-Myb-expressing breast tumors. Scientific Reports, Aug 2019, 9, 9.
Q1

ANGELUCCI, F., K. CECHOVA, M. VALIS, K. KUCA, et al. MicroRNAs in Alzheimer’s Disease: Diagnostic Markers or Therapeutic Agents? Frontiers in Pharmacology, Jun 2019, 10, 9.
Q1

LIGASOVA, A. AND K. KOBERNA Quantification of fixed adherent cells using a strong enhancer of the fluorescence of DNA dyes. Scientific Reports, Jun 2019, 9, 12.
Q1

NOVOSADOVA, E., Z. NAVRATILOVA, M. ORDELTOVA, M. ZURKOVA, et al. Comparison of lymphocyte immune phenotypes in bronchoalveolar lavage of non-smoking patients with sarcoidosis and other interstitial lung diseases. Journal of Thoracic Disease, Jun 2019, 11(6), 2287-+.
Q3

PELC, R., V. MASEK, V. LLOPIS-TORREGROSA, P. BOUR, et al. Spectral counterstaining in luminescence-enhanced biological Raman microscopy. Chemical Communications, Jul 2019, 55(57), 8329-8332.
Q1

STETKA, J., P. VYHLIDALOVA, L. LANIKOVA, P. KORALKOVA, et al. Addiction to DUSP1 protects JAK2V617F-driven polycythemia vera progenitors against inflammatory stress and DNA damage, allowing chronic proliferation. Oncogene, Jul 2019, 38(28), 5627-5642.
Q1

XAVIER, N. M., R. GONCALVES-PEREIRA, R. JORDA, D. HENDRYCHOVA, et al. Novel dodecyl-containing azido and glucuronamide-based nucleosides exhibiting anticancer potential. Pure and Applied Chemistry, Jul 2019, 91(7), 1085-1105.
Q2

JORDA, R., L. HAVLICEK, A. STURC, D. TUSKOVA, et al. 3,5,7-Substituted Pyrazolo 4,3-d pyrimidine Inhibitors of Cyclin-Dependent Kinases and Their Evaluation in Lymphoma Models. Journal of Medicinal Chemistry, May 2019, 62(9), 4606-4623.
Top 5

TURI, Z., M. LACEY, M. MISTRIK AND P. MOUDRY Impaired ribosome biogenesis: mechanisms and relevance to cancer and aging. Aging-Us, Apr 2019, 11(8), 2512-2540.
Q1

MAUGERI, A., J. HRUSKOVA, J. JAKUBIK, M. BARCHITTA, et al. Independent Effects of Hypertension and Obesity on Left Ventricular Mass and Geometry: Evidence from the Cardiovision 2030 Study. Journal of Clinical Medicine, Mar 2019, 8(3), 11.
Top 10

KRALOVA, P., S. BENICKA AND M. SOURAL Polymer-Assisted Synthesis of Single and Fused Diketomorpholines. Acs Combinatorial Science, Mar 2019, 21(3), 154-157.
Q2

TURNQUIST, C., J. A. BECK, I. HORIKAWA, I. E. OBIORAH, et al. Radiation-induced astrocyte senescence is rescued by Delta 133p53. Neuro-Oncology, Apr 2019, 21(4), 474-485.
Top 10

MARQUES, S. M., D. BEDNAR AND J. DAMBORSKY. Computational Study of Protein-Ligand Unbinding for Enzyme Engineering. Frontiers in Chemistry, Jan 2019, 6, 15.
Q2

MENSIKOVA, K., L. TUCKOVA, K. KOLARIKOVA, T. BARTONIKOVA, et al. Atypical parkinsonism of progressive supranuclear palsy-parkinsonism (PSP-P) phenotype with rare variants in FBXO7 and VPS35 genes associated with Lewy body pathology. Acta Neuropathologica, Jan 2019, 137(1), 171-173.
Top 5

SKODA, J., K. BORANKOVA, P. J. JANSSON, M. L. H. HUANG, et al. Pharmacological targeting of mitochondria in cancer stem cells: An ancient organelle at the crossroad of novel anti-cancer therapies. Pharmacological Research, Jan 2019, 139, 298-313.
Top 10

MUSIL, M., H. KONEGGER, J. HONG, D. BEDNAR, et al. Computational Design of Stable and Soluble Biocatalysts. Acs Catalysis, Feb 2019, 9(2), 1033-1054.
Top 10

POKORNA, A., P. BOBAL, M. ORAVEC, L. RAROVA, et al. Investigation of Permeation of Theophylline through Skin Using Selected Piperazine-2,5-Diones. Molecules, Feb 2019, 24(3), 14.
Q2

2018

HAKOBJANYAN, A., A. STAHELOVA, F. MRAZEK, J. PETRKOVA, et al. TP53 rs1042522 and rs8064946 variants in myocardial infarction. Bratislava Medical Journal-Bratislavske Lekarske Listy, 2018, 119(12), 747-751.
Q4

JORDA, R., D. HENDRYCHOVA, J. VOLLER, E. REZNICKOVA, et al. How Selective Are Pharmacological Inhibitors of Cell-Cycle-Regulating Cyclin-Dependent Kinases? Journal of Medicinal Chemistry, Oct 2018, 61(20), 9105-9120.
Top 5

LIGASOVA, A. AND K. KOBERNA DNA Replication: From Radioisotopes to Click Chemistry. Molecules, Nov 2018, 23(11), 18.
Q2